PMID | Article Title | Published | Deposition |
---|---|---|---|
31158743 | Caffeic acid phenethyl ester (CAPE)-derivatives act as selective inhibitors of acetylcholinesterase. | 01-SEP-2019 | 24-FEB-2021 |
30388464 | Computer-aided design, synthesis and biological characterization of novel inhibitors for PKMYT1. | 01-JAN-2019 | 19-FEB-2021 |
9461567 | Evidence for the absolute conformational specificity of the intestinal H+/peptide symporter, PEPT1. | 13-FEB-1998 | 30-AUG-2020 |
11284702 | A novel inhibitor of the mammalian peptide transporter PEPT1. | 10-APR-2001 | 30-AUG-2020 |
30220607 | Unexpected AChE inhibitory activity of (2E)?,?-unsaturated fatty acids. | 01-NOV-2018 | 18-AUG-2020 |
29941193 | Identification of PKMYT1 inhibitors by screening the GSK published protein kinase inhibitor set I and II. | 07-AUG-2018 | 17-AUG-2020 |
29494161 | Potent and Selective Inhibitors of Human Sirtuin 5. | 22-MAR-2018 | 15-DEC-2019 |
28478927 | Discovery of novel substituted benzo-anellated 4-benzylamino pyrrolopyrimidines as dual EGFR and VEGFR2 inhibitors. | 15-JUN-2017 | 15-OCT-2019 |
27936444 | Amino derivatives of platanic acid act as selective and potent inhibitors of butyrylcholinesterase. | 27-JAN-2017 | 18-JUN-2019 |
27689726 | Repurposing N,N'-bis-(arylamidino)-1,4-piperazinedicarboxamidines: An unexpected class of potent inhibitors of cholinesterases. | 05-JAN-2017 | 07-SEP-2018 |
26048803 | Discovery of substituted 1,4-dihydroquinolines as novel promising class of P-glycoprotein inhibitors: First structure-activity relationships and bioanalytical studies. | 13-JUN-2015 | 14-NOV-2016 |
24650640 | Discovery of 4-anilinoa-carbolines as novel Brk inhibitors. | 07-APR-2014 | 06-FEB-2015 |
22770610 | Evaluation of potential Myt1 kinase inhibitors by TR-FRET based binding assay. | 11-MAR-2013 | 24-SEP-2013 |
23039927 | Multitargeted drug development: Discovery and profiling of dihydroxy substituted 1-aza-9-oxafluorenes as lead compounds targeting Alzheimer disease relevant kinases. | 22-OCT-2012 | 17-MAY-2013 |
15974593 | Three-dimensional quantitative structure-activity relationship analyses of beta-lactam antibiotics and tripeptides as substrates of the mammalian H+/peptide cotransporter PEPT1. | 24-JUN-2005 | 03-DEC-2012 |
14667225 | Three-dimensional quantitative structure-activity relationship analyses of peptide substrates of the mammalian H+/peptide cotransporter PEPT1. | 11-DEC-2003 | 30-NOV-2012 |
12593668 | Evaluation of the first cytostatically active 1-aza-9-oxafluorenes as novel selective CDK1 inhibitors with P-glycoprotein modulating properties. | 20-FEB-2003 | 30-NOV-2012 |
22189141 | In vitro and in silico studies on substrate recognition and acceptance of human PKMYT1, a Cdk1 inhibitory kinase. | 13-JAN-2012 | 22-JUL-2012 |
21955456 | Three-dimensional quantitative structure-activity relationship analyses of substrates of the human proton-coupled amino acid transporter 1 (hPAT1). | 17-OCT-2011 | 21-JUL-2012 |
21035334 | Discovery and selectivity-profiling of 4-benzylamino 1-aza-9-oxafluorene derivatives as lead structures for IGF-1R inhibitors. | 08-NOV-2010 | 14-JUN-2011 |
10579836 | Synthesis and biological evaluation of the first N-alkyl cage dimeric 4-aryl-1,4-dihydropyridines as novel nonpeptidic HIV-1 protease inhibitors. | 17-DEC-1999 | 10-NOV-2009 |
16821788 | Structural requirements for the substrates of the H+/peptide cotransporter PEPT2 determined by three-dimensional quantitative structure-activity relationship analysis. | 06-JUL-2006 | 10-NOV-2009 |
16640345 | Biological evaluation of bishydroxymethyl-substituted cage dimeric 1,4-dihydropyridines as a novel class of p-glycoprotein modulating agents in cancer cells. | 27-APR-2006 | 10-NOV-2009 |
15664865 | Novel CDK inhibition profiles of structurally varied 1-aza-9-oxafluorenes. | 01-FEB-2005 | 30-JAN-2006 |